What are Non-Natural Amino Acids?
Why revolutionary? Natural amino acids limit what proteins can do. Non-natural ones add: fluorescent tags for imaging, bioorthogonal chemistry (reactions that work only in living cells), protease resistance (drugs last longer), metal binding for catalysis. Trastuzumab deruxtecan (2024 FDA) uses non-natural linkers - $2B+ market!
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📚 Glossary
🏆 Key Figures
Peter Schultz (2001-present)
Pioneered genetic code expansion, enabling site-specific incorporation of non-natural amino acids into proteins using engineered tRNA/synthetase pairs
Carolyn Bertozzi (2022 Nobel)
Nobel Prize in Chemistry 2022 for developing bioorthogonal chemistry - reactions that work inside living cells without disrupting biology
Morten Meldal (2022 Nobel)
Nobel Prize in Chemistry 2022 for independently discovering the copper-catalyzed azide-alkyne cycloaddition (CuAAC) click reaction
K. Barry Sharpless (2022 Nobel (2nd))
Coined 'click chemistry' concept and shared 2022 Nobel Prize (his second Nobel) for copper-catalyzed click chemistry
Jason Chin (2019)
Created the first synthetic organism (Syn61) with a fully recoded genome, freeing codons for expanded genetic code with non-natural amino acids
Kevan Shokat (2013-present)
Used non-natural amino acid chemistry to develop covalent drugs targeting KRAS G12C, a previously 'undruggable' cancer mutation